MS436

Overview

MS436 is a new class of bromodomain inhibitor, exhibits potent affinity of an estimated K i =30-50 nM for the BRD4 BrD1 and a 10-fold selectivity over the BrD2.

Application

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Product Information

• Catalog No.: HY-13959
• CAS No.: 1395084-25-9
• Molecular Formula: C18H17N5O3S
• Molecular Weight: 383.42
• Purity: 99.94%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 1 mg/mL (2.61 mM); Clear solution
• Availability: In-stock

Source

Original product source