GSK6853

Overview

GSK6853, a chemical probe, is a potent and selective inhibitor of the BRPF1 bromodomain . GSK6853 shows excellent BRPF1 potency ( pK d = 9.5) and greater than 1600-fold selectivity over all other bromodomains.

Application

Products | Products > Disease Areas > Cancer | Products > Disease Areas > Blood or Cardio-cerebrovascular Disease | Products > Disease Areas > Leukemia/Lymphoma/Myeloma | Products > Disease Areas > Blood Disease | Products > Signaling Pathways > Epigenetics | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > Epigenetic Reader Domain

Product Information

• Catalog No.: HY-100220
• CAS No.: 1910124-24-1
• Molecular Formula: C22H27N5O3
• Molecular Weight: 409.48
• Purity: 99.53%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (6.11 mM); Clear solution
• Availability: In-stock

Source

Original product source