MPO-IN-1

Overview

MPO-IN-1 is a potent, orally active, and irreversible indole-containing inhibitor of myeloperoxidase ( MPO ). MPO-IN-1 has IC 50 s of 2.6 μM and 5.3 μM for MPO and thyroid peroxidase (TPO), respectively. MPO-IN-1 inhibits MPO activity in an acute mouse model of inflammation.

Application

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Product Information

• Catalog No.: HY-139915
• CAS No.: 2471981-21-0
• Molecular Formula: C24H21ClN4
• Molecular Weight: 400.90
• Purity: 98.07%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 5 mg/mL (12.47 mM); Clear solution
• Availability: In-stock

Source

Original product source