MEK/PI3K-IN-2 (compound 6s) is a potent MEK/PI3K inhibitor, with IC 50 values of 352 nM ( MEK1 ), 107 nM ( PI3Kα ), and 137 nM ( PI3Kδ ), respectively. MEK/PI3K-IN-2 suppresses pAKT and pERK1/2 levels. MEK/PI3K-IN-2 shows anti-proliferative activity against tumor cell lines.
Products | Products > Signaling Pathways > MAPK/ERK Pathway | Products > Signaling Pathways > PI3K/Akt/mTOR | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > MEK | Products > Signaling Pathways > PI3K | Products > Signaling Pathways > PERK
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