CXCR2 antagonist 4 (compound 7) is a potent CXCR2 antagonist with an IC 50 value of 0.13 μM. CXCR2 antagonist 4 can inhibit CXCL8-induced cytosolic calcium increase (IC 50 = 27 μM). CXCR2 antagonist 4 can be used for researching anticancer .
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