Exarafenib

Overview

Exarafenib (RAF/KIN_2787) is an orally-available, selective pan- RAF inhibitor. Exarafenib is effective in RAF-dependent cancers, including all classes of BRAF alterations. Exarafenib suppresses MAPK signaling in RAF-dependent melanoma cell lines. Exarafenib has anticancer activity.

Application

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Product Information

• Catalog No.: HY-147268
• CAS No.: 2639957-39-2
• Molecular Formula: C26H34F3N5O3
• Molecular Weight: 521.58
• Purity: 99.77%
• Storage: 4°C, sealed storage, away from moisture and light * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
• Solubility: ≥ 2.5 mg/mL (4.79 mM); Clear solution
• Availability: In-stock

Source

Original product source