JNJ-6204 is a dual inhibitor for CSNK1D ( Casein Kinase 1 Delta) and CSNK1E ( Casein Kinase 1 Epsilon) (CSNK1D IC 50 =2.3 nM; CSNK1E IC 50 =137 nM). JNJ-6204 shows good brain exposure.
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