CGS 15943

Overview

CGS 15943 is an orally bioavailable non-xanthine Adenosine Receptor antagonist. Its K i for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM in transfected CHO cells, respectively. .

Application

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Product Information

• Catalog No.: HY-100678
• CAS No.: 104615-18-1
• Molecular Formula: C13H8ClN5O
• Molecular Weight: 285.69
• Purity: 99.55%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: 1.22 mg/mL (4.27 mM); Suspended solution; Need ultrasonic
• Availability: In-stock

Source

Original product source