LSD1-IN-26 (compound 12u) is a potent LSD1 inhibitor, with an IC 50 of 25.3 nM. LSD1-IN-26 also inhibits MAO-A ( IC 50 =1234.57 nM) and MAO-B ( IC 50 =3819.27 nM). LSD1-IN-26 significantly induces apoptosis in MGC-803 cells. LSD1-IN-26 can be used for gastric cancer research.
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