PBRM1-BD2-IN-7 is a selective and cell-active polybromo-1 (PBRM1) bromodomain inhibitor. PBRM1-BD2-IN-7 has inhibitory activity for PBRM1-BD2 with an IC 50 value of 0.29 μM. PBRM1-BD2-IN-7 can be used for the research of cancer .
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