PBRM1-BD2-IN-8

Overview

PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor (PBRM1-BD2 K d =4.4 μM, PBRM1-BD2 IC 50 =0.16 μM; PBRM1-BD5 K d =25 μM). PBRM1-BD2-IN-8 shows anti-cancer activity.

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Epigenetics | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Epigenetic Reader Domain | Products > Signaling Pathways > SWI/SNF Complex

Product Information

• Catalog No.: HY-151538
• CAS No.: 2819989-75-6
• Molecular Formula: C15H13BrN2O
• Molecular Weight: 317.18
• Purity: 98.05%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (7.88 mM); Clear solution
• Availability: In-stock

Source

Original product source