Polfurmetinib

Polfurmetinib
  • CAS No.:2845151-86-0
  • Grade:98.21%
  • Formula:C18H20FN3O4S
  • M.W.:393.43
  • Solvent:≥ 2.5 mg/mL (6.35 mM); Clear solution

Overview

Polfurmetinib (MEK-IN-6) (Example 69) is a MEK inhibitor. MEK-IN-6 inhibits ERK1/2 (Thr202/Tyr204) phosphorylation in A375 cells (IC 50 : 2 nM). Polfurmetinib can be used for research of cancer .

Application

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Product Information

  • Catalog No.: HY-153445
  • CAS No.: 2845151-86-0
  • Molecular Formula: C18H20FN3O4S
  • Molecular Weight: 393.43
  • Purity: 98.21%
  • Storage: Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
  • Solubility: ≥ 2.5 mg/mL (6.35 mM); Clear solution
  • Availability: In-stock

Source

Original product source


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