SOS1-IN-16 (Comp 54) is a selective inhibitor of SOS1 with an IC 50 of 7.2 nM. SOS1-IN-16 has inhibitory activity of CYP3A4 when using testosterone as a substrate, with an IC 50 of 8.9μM. SOS1-IN-16 can be used for cancer research.
Products | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Signaling Pathways > MAPK/ERK Pathway | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > Ras | Products > Signaling Pathways > SOS1 | Products > Signaling Pathways > Cytochrome P450
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