hCYP1B1-IN-1 (compound B18) is a hCYP1B1 inhibitor ( IC 50 =3.6 nM),as well as an antagonist of Aryl Hydrocarbon Receptor . hCYP1B1-IN-1 exhibtis suitable metabolic stability and good cell-permeability. hCYP1B1-IN-1 inhibits migration of MCF-7 cells.
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