CCT368772 (compound 35) is a selective kinesin HSET inhibitor ( HSET ADP-Glo IC 50 = 0.019 μM). CCT368772 exhibits selectivity over Eg5 ( Eg5 ADP-Glo IC 50 >200 μM). CCT368772 (compound 152) can be used for the study of hyperproliferative diseases and disorders such as cancer .
Products | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Signaling Pathways > Cytoskeleton | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Kinesin
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