JAK-IN-31 (Example 75) is a JAK inhibitor with IC 50 ranges of ≤0.01µM, ≤0.01µM, 0.01-0.1 µM and ≤0.01µM for JAK1 , JAK2 , JAK3 and Tyk2 respectively. JAK-IN-31 can be used in cancer research.
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