Afuresertib

Overview

Afuresertib (GSK2110183) is an orally bioavailable, selective, ATP-competitive and potent pan-Akt kinase inhibitor with K i s of 0.08/2/2.6 nM for Akt1/Akt2/Akt3, respectively.

Application

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Product Information

• Catalog No.: HY-15727
• CAS No.: 1047644-62-1
• Molecular Formula: C18H17Cl2FN4OS
• Molecular Weight: 427.32
• Purity: 99.53%
• Storage: -20°C, protect from light, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light, stored under nitrogen)
• Solubility: ≥ 2.5 mg/mL (5.85 mM); Clear solution
• Availability: In-stock

Source

Original product source