TEAD-IN-11 (compound 38) has a good inhibitory effect on TEAD1 ( IC 50 =8.7 nM), TEAD2 ( IC 50 =3.4 nM), TEAD3 ( IC 50 =5.6 nnM). TEAD-IN-11 has good selective activity against TEAD1-3 as a covalent inhibitor. TEAD-IN-11 can be used for cancer research.
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