JAK2/FLT3-IN-3 (11r) is a dual FLT3 and JAK2 inhibitor, with IC 50 values of 2.01 nM, 0.51 nM and 104.40 nM for JAK2 , FLT3 and JAK3 , respectively. JAK2/FLT3-IN-3 (11r) induces apoptosis and possesses antitumor activity.
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