C3TD879

Overview

C3TD879 is a Type I kinase inhibitor that potently inhibits CITK catalytic activity ( IC 50 = 12 nM). C3TD879 binds directly to full-length human CITK in cells (NanoBRET K d < 10 nM). C3TD879 is a chemical probe suitable for interrogating the complex biology of CITK.

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Immunotherapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Ser/Thr Protease

Product Information

• Catalog No.: HY-162266
• CAS No.: 2850259-33-3
• Molecular Formula: C22H28N4O
• Molecular Weight: 364.48
• Purity: 98.41%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (6.86 mM); Clear solution
• Availability: In-stock

Source

Original product source