α2A-AR agonist 1

Overview

α2A-AR agonist 1 (Compound B9) is a selective agonist for α2-adrenergic receptor ( α2A-AR ) with EC 50 of 0.23 nM. α2A-AR agonist 1 exhibits a hypnotic effect, with ED 50 of 0.138 mg/kg in the loss of righting reflex (LORR) experiment. α2A-AR agonist 1 exhibits metabolic stability in mouse liver microsomes.

Application

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Product Information

• Catalog No.: HY-162620
• CAS No.: 2971825-58-6
• Molecular Formula: C12H11BrN2O
• Molecular Weight: 279.13
• Purity: 99.92%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Availability: In-stock

Source

Original product source