MerTK/Axl-IN-1

Overview

MerTK/Axl-IN-1 (Compound A-910) is a potent and selective dual MerTK/Axl inhibitor, with IC 50 s of 4.2 and 8.8 nM in Ba/F3, and 0.2 and 0.9 nM in HTRF. MerTK/Axl-IN-1 results in pMerTK inhibition in vivo. MerTK/Axl-IN-1 has long half-life, high oral exposure and bioavailability.

Application

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Product Information

• Catalog No.: HY-162940
• CAS No.: 3036009-40-9
• Molecular Formula: C40H47FN6O4
• Molecular Weight: 694.84
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source