I-BET787

Overview

I-BET787 is a orally active BET bromine domain inhibitor with pIC 50 s of 7.1 and 5.9 for BRD4 BD1 and BRD4 BD2, respectively. I-BET787 has anti-inflammatory activity in mice.

Application

Products | Products > Disease Areas > Cancer | Products > Disease Areas > Blood or Cardio-cerebrovascular Disease | Products > Disease Areas > Inflammation or Immune System Disease | Products > Disease Areas > Leukemia/Lymphoma/Myeloma | Products > Disease Areas > Blood Disease | Products > Signaling Pathways > Epigenetics | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Inflammation/Immunology | Products > Signaling Pathways > Epigenetic Reader Domain

Product Information

• Catalog No.: HY-163729
• CAS No.: 2201082-98-4
• Molecular Formula: C16H20ClN3O2
• Molecular Weight: 321.80
• Purity: 99.88%
• Storage: RT, sealed storage, away from moisture and light. In solvent -80°C, 1 year , -20°C, 6 months
• Availability: In-stock

Source

Original product source