AGN-195183

Overview

AGN-195183 (IRX-5183) is a potent and selective agonist of RARα ( K d =3 nM) with improved binding selectivity relative to AGN 193836. AGN-195183 has no activity on RARβ/γ.

Application

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Product Information

• Catalog No.: HY-16684
• CAS No.: 367273-07-2
• Molecular Formula: C22H22ClF2NO4
• Molecular Weight: 437.86
• Purity: 99.75%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 1.1 mg/mL (2.51 mM); Clear solution
• Availability: In-stock

Source

Original product source