EPZ011989 hydrochloride

Overview

EPZ011989 hydrochloride is a potent and orally active Zeste Homolog 2 ( EZH2 ) inhibitor, with a K i value of <3 nM. EPZ011989 shows anti-tumor activity. EPZ011989 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

Application

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Product Information

• Catalog No.: HY-16986B
• CAS No.: 2095432-26-9
• Molecular Formula: C35H52ClN5O4
• Molecular Weight: 642.27
• Purity: 99.40%
• Storage: 4°C, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
• Solubility: 2.5 mg/mL (3.89 mM); Clear solution; Need ultrasonic
• Availability: In-stock

Source

Original product source