AS-254s

Overview

AS-254s is the inhibitor for absent, small, or homeotic-like 1 protein ( ASH1L ) with an IC 50 of 94 nM ( FP assay). AS-254s exhibits antiproliferative activity against MLL1-rearranged leukemic cells with GI 50 <1 μM. AS-254s induces the differentiation of MLL1-r leukemic cell.

Application

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Product Information

• Catalog No.: HY-170494
• CAS No.: 3096805-79-4
• Molecular Formula: C36H41ClN6O3S2
• Molecular Weight: 705.33
• Purity: 98.96%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (3.54 mM); Clear solution
• Availability: In-stock

Source

Original product source