UNC0737 is an orthosteric choline kinase inhibitor. UNC0737 is also a poor inhibitor of G9a ( IC 50 = 5000 nM) and GLP ( IC 50 > 10000 nM) in the SAHH-coupled assays.
Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Choline Kinase
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