DPP8/9-IN-2

Overview

DPP8/9-IN-2 (Compound 21) is a DPP8/9 inhibitor with IC 50 values of 0.22 nM and 3 nM, respectively, and K i values of 2.9 nM and 6 nM, respectively . DPP8/9-IN-2 has certain cardiotoxicity, with IC 50 values of 0.7 μM, 29.0 μM and 27.7 μM for hERG potassium channel , Nav1.5 sodium channel and Cav1.2 calcium channel , respectively. DPP8/9-IN-2 can be used in the research of diseases such as tumors.

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Dipeptidyl Peptidase | Products > Signaling Pathways > Calcium Channel | Products > Signaling Pathways > Sodium Channel | Products > Signaling Pathways > Potassium Channel

Product Information

• Catalog No.: HY-175226
• CAS No.: 3109603-86-0
• Molecular Formula: C30H30F3N3O2
• Molecular Weight: 521.57
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source