Intoplicine

Overview

Intoplicine (RP 60475), an antitumor derivative in the 7H-benzo[e]pyrido[4,3-b]indole series, is a DNA topoisomerase I and II inhibitor. Intoplicine strongly binds DNA (K A = 2 x 10 5 /M) and thereby increases the length of linear DNA.

Application

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Product Information

• Catalog No.: HY-101647
• CAS No.: 125974-72-3
• Molecular Formula: C21H24N4O
• Molecular Weight: 348.44
• Purity: 98.36%
• Storage: 4°C, sealed storage, away from moisture and light * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
• Solubility: ≥ 2 mg/mL (5.74 mM); Clear solution
• Availability: In-stock

Source

Original product source