OPN-9643

Overview

OPN-9643 is a covalent inhibitor targeting the central palmitate binding pocket of TEADs with an IC 50 of 15 nM, preventing autopalmitoylation and reducing TEAD -driven luciferase activity and canonical TEAD targets, CTGF and CYR61 . OPN-9643 can be used for the research of cancer , such as melanoma.

Application

Products | Products > Disease Areas > Cancer | Products > Disease Areas > Melanoma | Products > Signaling Pathways > Stem Cell/Wnt | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Stem Cells | Products > Signaling Pathways > YAP

Product Information

• Catalog No.: HY-179559
• CAS No.: 2866423-06-3
• Molecular Formula: C19H16F3NO2
• Molecular Weight: 347.33
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source