GRPR antagonist-3

Overview

GRPR antagonist-3 (compound (S)-1m) is a potent GRPR antagonist with an IC 50 of 121 nM. GRPR antagonist-3 is stable in rat plasma and towards microsomal oxidative metabolism in vitro. GRPR antagonist-3 can be radiolabeled with fluorine-18 for PET imaging.

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > GPCR/G Protein | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Bombesin Receptor

Product Information

• Catalog No.: HY-180434
• CAS No.: 2077238-49-2
• Molecular Formula: C33H37FN6O5
• Molecular Weight: 616.68
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source