CHI3L1-IN-6 (Compound 9e) is a CHI3L1 inhibitor with a K d of 19.11 μM for hCHI3L1. CHI3L1-IN-6 blocks CHI3L1- Galectin-3 interaction. CHI3L1-IN-6 reduces STAT3 signaling. CHI3L1-IN-6 exhibits anti-cancer activity against glioblastoma.
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