Filgotinib-d 4

Filgotinib-d 4
  • CAS No.:2041095-50-3
  • Grade:99.98%
  • Formula:C21H19D4N5O3S
  • M.W.:429.53

Overview

Filgotinib-d 4 is the deuterium labeled Filgotinib. Filgotinib (GLPG0634) is a selective JAK1 inhibitor with IC50 of 10 nM, 28 nM, 810 nM, and 116 nM for JAK1 , JAK2 , JAK3 , and TYK2 , respectively.

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Epigenetics | Products > Signaling Pathways > Stem Cell/Wnt | Products > Signaling Pathways > Protein Tyrosine Kinase/RTK | Products > Signaling Pathways > JAK/STAT Signaling | Products > Research Areas > Cancer > Cancer Stem Cells | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > JAK

Product Information

  • Catalog No.: HY-18300S
  • CAS No.: 2041095-50-3
  • Molecular Formula: C21H19D4N5O3S
  • Molecular Weight: 429.53
  • Purity: 99.98%
  • Storage: Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
  • Availability: In-stock

Source

Original product source


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