Numidargistat dihydrochloride

Overview

Numidargistat (CB-1158) dihydrochloride is a potent and orally active inhibitor of arginase , with IC 50 s of 86 nM and 296 nM for recombinant human arginase 1 and recombinant human arginase 2 , respectively. Immuno-oncology agent.

Application

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Product Information

• Catalog No.: HY-101979A
• CAS No.: 2095732-06-0
• Molecular Formula: C11H24BCl2N3O5
• Molecular Weight: 360.04
• Purity: 98.50%
• Storage: -20°C, stored under nitrogen, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen, away from moisture)
• Solubility: 3.25 mg/mL (9.03 mM); Suspended solution; Need ultrasonic
• Availability: In-stock

Source

Original product source