INCB3344

Overview

INCB3344 is a potent, selective and orally bioavailable CCR2 antagonist with IC 50 values of 5.1 nM (hCCR2) and 9.5 nM (mCCR2) in binding antagonism and 3.8 nM (hCCR2) and 7.8 nM (mCCR2) in antagonism of chemotaxis activity.

Application

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Product Information

• Catalog No.: HY-50674
• CAS No.: 1262238-11-8
• Molecular Formula: C29H34F3N3O6
• Molecular Weight: 577.59
• Purity: 99.81%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: 6 mg/mL (10.39 mM); Clear solution; Need ultrasonic
• Availability: In-stock

Source

Original product source