cis-INCB3344

Overview

cis-INCB3344 is the isomer of INCB3344 ( HY-50674 ), and can be used as an experimental control. INCB3344 is a potent, selective and orally bioavailable CCR2 antagonist with IC 50 values of 5.1 nM (hCCR2) and 9.5 nM (mCCR2) in binding antagonism and 3.8 nM (hCCR2) and 7.8 nM (mCCR2) in antagonism of chemotaxis activity.

Application

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Product Information

• Catalog No.: HY-77111
• CAS No.: 1285539-85-6
• Molecular Formula: C29H34F3N3O6
• Molecular Weight: 577.59
• Purity: 95.10%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Availability: In-stock

Source

Original product source