Perphenazine is an orally active dopamine receptor and histamine-1 receptor antagonist, with K i values of 0.56 nM (D2), 0.43 nM (D3), 6 nM (5-HT2A), respectively. Perphenazine also binds to Alpha-1A adrenergic receptor . Perphenazine inhibits cancer cell proliferation, and induces apoptosis . Perphenazine can be used in the research of mental disease, cancer , inflammation.
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