Mosapride citrate is an orally active gastroenterokinetic compound. Mosapride citrate is a 5HT4 agonist. Mosapride citrate is a CYP inducer. Mosapride citrate has a concentration-dependent inhibitory effect on Kv4.3 , and its IC 50 value is 15.2 μM. Mosapride citrate can be used in the study of gastrointestinal diseases.
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