Palupiprant

Overview

Palupiprant (E7046) is an orally bioavailable and specific EP4 antagonist, with IC 50 of 13.5 nM and K i of 23.14 nM. Palupiprant exhibits anti-tumor activities.

Application

Products | Products > Disease Areas > Cancer | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Endocrinology | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Immunotherapy | Products > Signaling Pathways > Prostaglandin Receptor

Product Information

• Catalog No.: HY-103088
• CAS No.: 1369489-71-3
• Molecular Formula: C22H18F5N3O4
• Molecular Weight: 483.39
• Purity: 99.96%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.08 mg/mL (4.30 mM); Clear solution
• Availability: In-stock

Source

Original product source