Epinastine hydrochloride

Overview

Epinastine hydrochloride (WAL801 hydrochloride) is a selective and orally active histamine H1 receptor antagonist, CD96/PVR inhibitor and mast cell stabilizer. Epinastine hydrochloride has high affinity for neuronal octopamine receptors in locusts ( K i = 2 nM) and honeybees ( K i = 1.1 nM). Epinastine hydrochloride inhibits TARC , IL-8 , and IL-4 . Epinastine hydrochloride activates anti-colon cancer immunity and inhibits Substance P ( HY-P0201 )-induced scratching behavior and increased vascular permeability. Epinastine hydrochloride can be used in the research of allergic diseases.

Application

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Product Information

• Catalog No.: HY-B0640A
• CAS No.: 108929-04-0
• Molecular Formula: C16H16ClN3
• Molecular Weight: 285.77
• Purity: 99.86%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.08 mg/mL (7.28 mM); Clear solution
• Availability: In-stock

Source

Original product source