CGP 57380

Overview

CGP 57380 is a cell-permeable pyrazolo-pyrimidine compound that acts as a selective inhibitor of Mnk1 with IC 50 of 2.2 μM, but has no inhibitory activity against p38, JNK1 , ERK1/2, PKC , or Src-like kinases.

Application

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Product Information

• Catalog No.: HY-10520
• CAS No.: 522629-08-9
• Molecular Formula: C11H9FN6
• Molecular Weight: 244.23
• Purity: 98.71%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (10.24 mM); Clear solution
• Availability: In-stock

Source

Original product source