Golidocitinib

Overview

Golidocitinib (AZD4205) is a selective JAK1 inhibitor, with an IC 50 of 73 nM, weakly inhibits JAK2 ( IC 50 >14.7 μM), and shows little inhibition on JAK3 ( IC 50 >30 μM).

Application

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Product Information

• Catalog No.: HY-107361
• CAS No.: 2091134-68-6
• Molecular Formula: C25H31N9O2
• Molecular Weight: 489.57
• Purity: 99.54%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (5.11 mM); Clear solution
• Availability: In-stock

Source

Original product source