PDK1-IN-1 (Compound 2-11) is a PDK1 inhibitor. PDK1-IN-1 is also useful as inhibitor of other kinases such as FGFR3 , NTRK3 , RP-S6K and WEE1 . PDK1-IN-1 selectively inhibits microtubule affinity regulating kinase ( MARK ). PDK1-IN-1 can be used for researches of myeloproliferative disorders, cancer and Alzheimer's disease.
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